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Cayman 1-Deoxynojirimycin (Hydrochloride); Purity- Greater Than O
Cayman 1-Deoxynojirimycin (Hydrochloride); Purity- Greater Than Or Equal To 95%; Size- 5 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
List Price
$33.00
Your Price
$33.00
HOW MUCH YOU SAVE:
0.00 %
NETA PART: | CAYM-10011718-5 |
MFG.PART: | 10011718-5 |
UNSPSC: | 12352200 |
Manufacturer: | Cayman |
Product Description
ICA 121431 is a voltage-gated sodium channel (Nav) blocker that selectively blocks Nav1.1 and Nav1.3 over Nav1.4, and Nav1.5-1.8 channels (IC50s = <20, 19, 240, and >10,000 nM, respectively). It induces a concentration-dependent hyperpolarizing shift in voltage dependence of inactivation of Nav1.3 channels at a concentration 1 μM but has no effect on resting channels. Substitution of the Nav1.3 domain IV voltage-sensor domain (VSD4) with the Nav1.5 VSD4 reduces ICA 121431 potency by approximately 500-fold.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
α-phenyl-N- [4-[(2-thiaz olylamino) sulfonyl] phenyl]- benzene acetamide
CAS Number
313254-51-2
Molecular Formula
C23H19N3O3S2
Formula Weight
449.5
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 15 mg/ml
- DMSO: 15 mg/ml
- DMSO:PBS (pH 7.2) (1:1): 0.5 mg/ml
- Ethanol: 0.1 mg/ml
λmax
205, 260, 287 nm
SMILES
O=C(NC1=CC=C(S(NC2=NC=CS2)(=O)=O)C=C1)C(C3=CC=CC=C3)C4=CC=CC=C4
InChi Code
InChI=1S/C23H19N3O3S2/c27-22(21(17-7-3-1-4-8-17)18-9-5-2-6-10-18)25-19-11-13-20(14-12-19)31(28,29)26-23-24-15-16-30-23/h1-16,21H,(H,24,26)(H,25,27)
InChi Key
URSQNPPONHUJDL-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
SKU | CAYM-10011718-5 |
---|---|
Supplier Part Number | 10011718-5 |
UM | UNIT |
UNSPSC | 12352200 |
Manufacturer | Cayman |
MSDS URL | https://www.caymanchem.com/msdss/10011718m.pdf |
Temperature | -20 |
Refrigerated-Frozen | Refrigerated |
CountryOfOrigin | US |
ProductLine | CAYM |
Qty | 5 |
MinOrderQty | 1 |
Weight | 7.00 |
Lead Time | 2 Business Days |
Hazardous | N |
CAS Number | 73285-50-4 |