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Cayman Ha-130; Purity- Greater Than Or Equal To 98%; Size- 10 Mg
Cayman Ha-130; Purity- Greater Than Or Equal To 98%; Size- 10 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
List Price
$129.00
Your Price
$129.00
HOW MUCH YOU SAVE:
0.00 %
NETA PART: | CAYM-10498-10 |
MFG.PART: | 10498-10 |
UNSPSC: | 12352200 |
Manufacturer: | Cayman |
Product Description
HA-130 is a reversible inhibitor of autotaxin, completely blocking the hydrolysis of the substrate bis-pNPP with an IC50 value of 28 nM. It does not affect the activity of any proteasomal protease or related enzymes. HA-130 rapidly decreases plasma lysophosphatidic acid levels in mice when given intravenously (1 nM/g). HA-130 has been used to investigate the role of autotaxin in cells and animals.,,
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
B- [3- [[4- [[3- [(4- fluorophenyl)methyl]- 2,4- dioxo- 5- thiazolidinylidene]methyl]phenoxy]methyl]phenyl]- boronic acid
CAS Number
1229652-21-4
Molecular Formula
C24H19BFNO5S
Formula Weight
463.3
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 10 mg/mL
- DMSO: 5 mg/mL
- Ethanol: 0.5 mg/mL
λmax
239, 348 nm
SMILES
FC1=CC=C(CN2C(/C(SC2=O)=C/C3=CC=C(OCC4=CC=CC(B(O)O)=C4)C=C3)=O)C=C1
InChi Code
InChI=1S/C24H19BFNO5S/c26-20-8-4-17(5-9-20)14-27-23(28)22(33-24(27)29)13-16-6-10-21(11-7-16)32-15-18-2-1-3-19(12-18)25(30)31/h1-13,30-31H,14-15H2/b22-13-
InChi Key
VTNKMYWFWQTEHE-XKZIYDEJSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
SKU | CAYM-10498-10 |
---|---|
Supplier Part Number | 10498-10 |
UM | EA |
UNSPSC | 12352200 |
Manufacturer | Cayman |
MSDS URL | https://www.caymanchem.com/msdss/10498m.pdf |
Temperature | -20 |
Refrigerated-Frozen | Refrigerated |
CountryOfOrigin | CN |
ProductLine | CAYM |
Qty | 1 |
MinOrderQty | 1 |
Weight | 7.00 |
Lead Time | 2 Business Days |
Hazardous | N |
CAS Number | 1229652-21-4 |