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Cayman 9(S)-Pahsa; Purity- Greater Than Or Equal To 95%; Size- 1
Cayman 9(S)-Pahsa; Purity- Greater Than Or Equal To 95%; Size- 1 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
List Price
$576.00
Your Price
$576.00
HOW MUCH YOU SAVE:
0.00 %
NETA PART: | CAYM-18023-1 |
MFG.PART: | 18023-1 |
UNSPSC: | 12352200 |
Manufacturer: | Cayman |
Product Description
EX-527 is an inhibitor of sirtuin 1 (SIRT1; IC50 = 0.098 µM). It is selective for SIRT1 over SIRT2, and SIRT3 (IC50s = 19.6 and 48.7 µM, respectively) and the cytochrome P450 (CYP) isoforms CYP3A4, CYP2D6, CYP2C9, CYP2C19, and CYP1A2 at 1 µM. EX-527 (50 µM) induces cell cycle arrest at the G1 phase in MCF-7 cells.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
6-chloro- 2,3,4,9- tetrahydro- 1H-carbazole- 1-carboxamide
CAS Number
49843-98-3
Molecular Formula
C13H13ClN2O
Formula Weight
248.7
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 20 mg/ml
- DMSO: 20 mg/ml
- DMSO:PBS(pH7.2) (1:1): 0.5 mg/ml
- Ethanol: 5 mg/ml
λmax
233, 291 nm
SMILES
ClC(C=C1)=CC2=C1NC3=C2CCCC3C(N)=O
InChi Code
InChI=1S/C13H13ClN2O/c14-7-4-5-11-10(6-7)8-2-1-3-9(13(15)17)12(8)16-11/h4-6,9,16H,1-3H2,(H2,15,17)
InChi Key
FUZYTVDVLBBXDL-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
SKU | CAYM-18023-1 |
---|---|
Supplier Part Number | 18023-1 |
UM | UNIT |
UNSPSC | 12352200 |
Manufacturer | Cayman |
MSDS URL | https://www.caymanchem.com/msdss/18023m.pdf |
Temperature | -20 |
Refrigerated-Frozen | Refrigerated |
CountryOfOrigin | US |
ProductLine | CAYM |
Qty | 1 |
MinOrderQty | 1 |
Weight | 7.00 |
Lead Time | 2 Business Days |
Hazardous | Y |
CAS Number | 2097130-87-3 |