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Cayman Ylf-466d; Purity- Greater Than Or Equal To 98%; Size- 5 Mg
Cayman Ylf-466d; Purity- Greater Than Or Equal To 98%; Size- 5 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
List Price
$467.00
Your Price
$467.00
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| NETA PART: | CAYM-19475-5 |
| MFG.PART: | 19475-5 |
| UNSPSC: | 12352200 |
| Manufacturer: | Cayman |
Product Description
Orphenadrine is a muscarinic acetylcholine receptor (mAChR) antagonist (Kds = 48, 213, 120, 170, and 129 nM for M1-M5 receptors, respectively). Orphenadrine (2-5 mg/kg, i.v.) decreases muscle activity induced by the mAChR agonist oxotremorine in rabbits. It is also an NMDA receptor antagonist with a Ki value of 6 µM in a radioligand binding assay in human postmortem frontal cortex and an IC50 value of 16.2 µM for inhibiting steady state currents in cultured superior colliculus neurons. Formulations containing orphenadrine have been used in the treatment of acute painful musculoskeletal conditions, including muscle spasms.
WARNING This product is not for human or veterinary use.
Technical Information
| Formal Name | N,N-dimethyl-2-[(2-methylphenyl)phenylmethoxy]-ethanamine, monohydrochloride |
| CAS Number | 341-69-5 |
| Synonyms |
|
| Molecular Formula | C18H23NO • HCl |
| Formula Weight | 305.8 |
| Purity | ≥98% |
| Formulation | A crystalline solid |
| Solubility |
|
| SMILES | CN(C)CCOC(C1=CC=CC=C1C)C2=CC=CC=C2.Cl |
| InChi Code | InChI=1S/C18H23NO.ClH/c1-15-9-7-8-12-17(15)18(20-14-13-19(2)3)16-10-5-4-6-11-16;/h4-12,18H,13-14H2,1-3H3;1H |
| InChi Key | UQZKYYIKWZOKKD-UHFFFAOYSA-N |
| Storage | -20°C |
| Shipping | Room Temperature in continental US; may vary elsewhere |
| Stability | ≥ 4 years |
| SKU | CAYM-19475-5 |
|---|---|
| Supplier Part Number | 19475-5 |
| UM | UNIT |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | https://www.caymanchem.com/msdss/19475m.pdf |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| CountryOfOrigin | US |
| ProductLine | CAYM |
| Qty | 5 |
| MinOrderQty | 1 |
| Weight | 7.00 |
| Lead Time | 2 Business Days |
| Hazardous | N |
| CAS Number | 1273323-67-3 |