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Cayman Ljh685; Purity- Greater Than Or Equal To 98%; Size- 1 Mg;
Cayman Ljh685; Purity- Greater Than Or Equal To 98%; Size- 1 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
List Price
$32.00
Your Price
$32.00
HOW MUCH YOU SAVE:
0.00 %
NETA PART: | CAYM-19913-1 |
MFG.PART: | 19913-1 |
UNSPSC: | 12352200 |
Manufacturer: | Cayman |
Product Description
GSK1292263 is an agonist of G protein-coupled receptor 119 (GPR119; EC50 = 43.9 nM in CHO-K1 cells expressing human receptors). It inhibits increases in sterol regulatory element binding protein-1 (SREBP-1) levels induced by the LXR agonist T0901317 and increases activation of AMPK in HepG2 cells in a concentration-dependent manner. GSK1292263 also inhibits breast cancer resistant protein (BCRP) and organic anion transporting polypeptide 1B1 (OATP1B1) by 52 and 40%, respectively, when used at a concentration of 3 μM.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
5-[[1-[3-(1- methylethyl)- 1,2,4- oxadiazol-5- yl]-4- piperidinyl] methoxy]-2- [4-(methyl sulfonyl) phenyl]- pyridine
CAS Number
1032823-75-8
Molecular Formula
C23H28N4O4S
Formula Weight
456.6
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMSO: 30 mg/mL
λmax
224, 276, 296 nm
SMILES
CS(C1=CC=C(C2=CC=C(OCC3CCN(C4=NC(C(C)C)=NO4)CC3)C=N2)C=C1)(=O)=O
InChi Code
InChI=1S/C23H28N4O4S/c1-16(2)22-25-23(31-26-22)27-12-10-17(11-13-27)15-30-19-6-9-21(24-14-19)18-4-7-20(8-5-18)32(3,28)29/h4-9,14,16-17H,10-13,15H2,1-3H3
InChi Key
AYJRTVVIBJSSKN-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
SKU | CAYM-19913-1 |
---|---|
Supplier Part Number | 19913-1 |
UM | UNIT |
UNSPSC | 12352200 |
Manufacturer | Cayman |
MSDS URL | https://www.caymanchem.com/msdss/19913m.pdf |
Temperature | -20 |
Refrigerated-Frozen | Refrigerated |
CountryOfOrigin | CN |
ProductLine | CAYM |
Qty | 1 |
MinOrderQty | 1 |
Weight | 7.00 |
Lead Time | 2 Business Days |
Hazardous | N |
CAS Number | 1627710-50-2 |