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Cayman Andrastin A; Purity- Greater Than Or Equal To 95%; Size- 5
Cayman Andrastin A; Purity- Greater Than Or Equal To 95%; Size- 500 Micrograms; - CAYM (Additional S&H Or Hazmat Fees May Apply)
List Price
$211.05
Your Price
$211.05
HOW MUCH YOU SAVE:
0.00 %
| NETA PART: | CAYM-22067-500 |
| MFG.PART: | 22067-500 |
| UNSPSC: | 12352200 |
| Manufacturer: | Cayman |
Product Description
Cisapride is an agonist of serotonin (5-HT) receptor subtype 5-HT4 (IC50 = 0.483 μM in COS-7 cells expressing the human receptor). It induces relaxation of precontracted isolated rat esophageal thoracic muscularis mucosae preparations (EC50 = 102.33 nM). Cisapride (0.5 mg/kg) increases the rate of gastric emptying in rats. It is also a human ether-a-go-go related gene (hERG) channel blocker that binds to hERG channels with an IC50 value of less than 1 μM in a fluorescence polarization assay. Formulations containing cisapride have previously been used in the treatment of nocturnal heartburn associated with gastroesophageal reflux disease.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
rel-4-amino-5
CAS Number
81098-60-4
Molecular Formula
C23H29ClFN3O4
Formula Weight
466.0
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 30 mg/ml
- DMSO: 30 mg/ml
- DMSO:PBS (pH 7.2) (1:4): 0.2 mg/ml
- Ethanol: slightly soluble
λmax
214, 276, 308 nm
SMILES
NC1=CC(OC)=C(C(N[C@@H]2CCN(CCCOC3=CC=C(F)C=C3)C[C@@H]2OC)=O)C=C1Cl
InChi Code
InChI=1S/C23H29ClFN3O4/c1-30-21-13-19(26)18(24)12-17(21)23(29)27-20-8-10-28(14-22(20)31-2)9-3-11-32-16-6-4-15(25)5-7-16/h4-7,12-13,20,22H,3,8-11,14,26H2,1-2H3,(H,27,29)/t20-,22+/m1/s1
InChi Key
DCSUBABJRXZOMT-IRLDBZIGSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-22067-500 |
|---|---|
| Supplier Part Number | 22067-500 |
| UM | UNIT |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | https://www.caymanchem.com/msdss/22067m.pdf |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| CountryOfOrigin | AU |
| ProductLine | CAYM |
| Qty | 500 |
| MinOrderQty | 1 |
| Weight | 7.00 |
| Lead Time | 2 Business Days |
| Hazardous | N |
| CAS Number | 174232-42-9 |