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Cayman Calpain Inhibitor Vi; Purity- Greater Than Or Equal To 95%
Cayman Calpain Inhibitor Vi; Purity- Greater Than Or Equal To 95%; Size- 1 Mg; - CAYM (Additional S&H Or Hazmat Fees May Apply)
List Price
$73.00
Your Price
$73.00
HOW MUCH YOU SAVE:
0.00 %
NETA PART: | CAYM-23942-1 |
MFG.PART: | 23942-1 |
UNSPSC: | 12352200 |
Manufacturer: | Cayman |
Product Description
Mycophenolic acid β-D-glucuronide (MPAG) is a metabolite of the immunosuppressant mycophenolic acid (Item No. )., It is formed from mycophenolic acid by the UDP-glucuronosyltransferase (UGT) isoforms UGT1A9, UGT1A8, UGT1A7, and UGT1A10 in insect cell-derived supersomes expressing the human enzymes. Unlike mycophenolic acid, MPAG does not inhibit IMP dehydrogenase (IMPDH) type II in a cell-free assay. However, it does reduce tumor growth in an Ehrlich murine spontaneous adenocarcinoma model when administered at a dose of 6 mg/animal.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
5-[(2E)-5-carboxy- 3-methyl-2-penten-1-yl]- 1,3-dihydro-6-methoxy- 7-methyl-3-oxo-4- isobenzofuranyl β-D-glucopyranosiduronic acid
CAS Number
31528-44-6
Synonyms
- MPAG
- MPA-phenyl-glucuronide
- Mycophenolic Acid Glucosiduronate
Molecular Formula
C23H28O12
Formula Weight
496.5
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 5 mg/ml
- DMSO: 10 mg/ml
- PBS (pH 7.2): 10 mg/ml
λmax
214, 250, 292 nm
SMILES
O=C1OCC2=C(C)C(OC)=C(C/C=C(C)/CCC(O)=O)C(O[C@@H]3O[C@H](C(O)=O)[C@@H](O)[C@H](O)[C@H]3O)=C21
InChi Code
InChI=1S/C23H28O12/c1-9(5-7-13(24)25)4-6-11-18(32-3)10(2)12-8-33-22(31)14(12)19(11)34-23-17(28)15(26)16(27)20(35-23)21(29)30/h4,15-17,20,23,26-28H,5-8H2,1-3H3,(H,24,25)(H,29,30)/b9-4+/t15-,16-,17+,20-,23+/m0/s1
InChi Key
BYFGTSAYQQIUCN-HGIHDBQLSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
SKU | CAYM-23942-1 |
---|---|
Supplier Part Number | 23942-1 |
UM | UNIT |
UNSPSC | 12352200 |
Manufacturer | Cayman |
MSDS URL | https://www.caymanchem.com/msdss/23942m.pdf |
Temperature | -20 |
Refrigerated-Frozen | Refrigerated |
CountryOfOrigin | US |
ProductLine | CAYM |
Qty | 1 |
MinOrderQty | 1 |
Weight | 7.00 |
Lead Time | 2 Business Days |
Hazardous | N |
CAS Number | 190274-53-4 |