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Cayman Vs-5584 Analog
Cayman Vs-5584 Analog - CAYM (Additional S&H Or Hazmat Fees May Apply)
List Price
$193.00
Your Price
$193.00
HOW MUCH YOU SAVE:
0.00 %
| NETA PART: | CAYM-30324-5 |
| MFG.PART: | 30324-5 |
| UNSPSC: | 12352200 |
| Manufacturer: | Cayman |
Product Description
Mepyramine is a first generation antihistamine that acts as an inverse agonist at the histamine H1 receptor. It is reported to bind with high affinity to a Gq/11 protein-coupled form of the receptor and to promote a G protein-coupled inactive state of the H1 receptor that interferes with the Gq/11-mediated signaling of the endogenously expressed receptor, as well as to reduce G protein availability for other non-related receptors associated with this signaling pathway. Mepyramine has been shown to inhibit histamine-induced inositol phosphate production with a log EC50 value of -7.94.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
N1-[(4-methox
CAS Number
59-33-6
Synonyms
- NSC 3604
- Pyrilamine
Molecular Formula
C17H23N3O • C4H4O4
Formula Weight
401.5
Purity
≥95%
Formulation
A crystalline solid
Solubility
- DMF: 25 mg/ml
- DMSO: 20 mg/ml
- Ethanol: 20 mg/ml
- PBS (pH 7.2): 10 mg/ml
λmax
245, 306 nm
SMILES
COC(C=C1)=CC=C1CN(CCN(C)C)C2=NC=CC=C2.OC(/C=C\C(O)=O)=O
InChi Code
InChI=1S/C17H23N3O.C4H4O4/c1-19(2)12-13-20(17-6-4-5-11-18-17)14-15-7-9-16(21-3)10-8-15;5-3(6)1-2-4(7)8/h4-11H,12-14H2,1-3H3;1-2H,(H,5,6)(H,7,8)/b;2-1-
InChi Key
JXYWFNAQESKDNC-BTJKTKAUSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-30324-5 |
|---|---|
| Supplier Part Number | 30324-5 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | https://www.caymanchem.com/msdss/30324m.pdf |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| CountryOfOrigin | CN |
| ProductLine | CAYM |
| Qty | 5 |
| MinOrderQty | 1 |
| Weight | 7.00 |
| Lead Time | 2 Business Days |
| Hazardous | N |
| CAS Number | 1246535-95-4 |