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Cayman Tianeptine-D6 (Hydrochloride)
Cayman Tianeptine-D6 (Hydrochloride) - CAYM (Additional S&H Or Hazmat Fees May Apply)
List Price
$481.00
Your Price
$481.00
HOW MUCH YOU SAVE:
0.00 %
| NETA PART: | CAYM-36800-1 |
| MFG.PART: | 36800-1 |
| UNSPSC: | 12352200 |
| Manufacturer: | Cayman |
Product Description
PSB-12379 is an inhibitor of ecto-5’-nucleotidase (CD73; Kis = 2.21 and 9.03 nM for the recombinant human and rat enzyme, respectively). It is selective for CD73 over human nucleoside triphosphate diphosphohydrolase 1 (NTPDase 1), -2, and -3, ectonucleotide pyrophosphatase/phosphodiesterase family member 1 (ENPP1), -2, and -3 (Kis = >10,000 nM for all), as well as the purinergic P2Y1 and P2Y12 receptors at 10 µM. PSB-12379 inhibits CD73 in isolated human serum with a Ki value of 18.8 nM.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
N-(phenylmethyl)-
CAS Number
1802226-78-3
Molecular Formula
C18H23N5O9P2
Formula Weight
515.4
Purity
≥98%
Formulation
A solid
Solubility
- Water: 5 mg/ml, sonicated
SMILES
O=P(CP(O)(O)=O)(O)OC[C@@H]1[C@@H](O)[C@@H](O)[C@]([H])(N2C=NC3=C(NCC4=CC=CC=C4)N=CN=C32)O1
InChi Code
InChI=1S/C18H23N5O9P2/c24-14-12(7-31-34(29,30)10-33(26,27)28)32-18(15(14)25)23-9-22-13-16(20-8-21-17(13)23)19-6-11-4-2-1-3-5-11/h1-5,8-9,12,14-15,18,24-25H,6-7,10H2,(H,29,30)(H,19,20,21)(H2,26,27,28)/t12-,14-,15-,18-/m1/s1
InChi Key
DMBYYIJBPDWQFF-SCFUHWHPSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-36800-1 |
|---|---|
| Supplier Part Number | 36800-1 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| MSDS URL | https://www.caymanchem.com/msdss/36800m.pdf |
| Temperature | -20 |
| Refrigerated-Frozen | Refrigerated |
| CountryOfOrigin | CA |
| ProductLine | CAYM |
| Qty | 1 |
| MinOrderQty | 1 |
| Weight | 7.00 |
| Lead Time | 2 Business Days |
| Hazardous | N |