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Cayman Bph-1358; 5 Mg; 5352-53-4; ≥95%
Cayman Bph-1358; 5 Mg; 5352-53-4; ≥95% - CAYM (Additional S&H Or Hazmat Fees May Apply)
List Price
$79.00
Your Price
$79.00
HOW MUCH YOU SAVE:
0.00 %
NETA PART: | CAYM-37402-5 |
MFG.PART: | 37402-5 |
UNSPSC: | 12352200 |
Manufacturer: | Cayman |
Product Description
Mps1-IN-2 is an ATP-competitive inhibitor of the checkpoint kinase Mps1 (IC50 = 145 nM). It is 1,000-fold selective for Mps1 over a panel of 352 kinases at 10 μM, but does inhibit Plk1 (Kd = 61 nM).
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
9-cyclopentyl- 2-[[2-ethoxy- 4-(4-hydroxy- 1-piperidinyl)phenyl]amino]- 5,7,8,9-tetrahydro- 5-methyl- 6H-pyrimido[4,5-b][1,4]diazepin- 6-one
CAS Number
1228817-38-6
Molecular Formula
C26H36N6O3
Formula Weight
480.6
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 1 mg/ml
- DMF:PBS (pH 7.2)(1:3): 0.25 mg/ml
- DMSO: 1 mg/ml
- Ethanol: slightly soluble
λmax
288 nm
SMILES
OC1CCN(C2=CC(OCC)=C(NC3=NC=C(N(C)C(CCN4C5CCCC5)=O)C4=N3)C=C2)CC1
InChi Code
InChI=1S/C26H36N6O3/c1-3-35-23-16-19(31-13-10-20(33)11-14-31)8-9-21(23)28-26-27-17-22-25(29-26)32(18-6-4-5-7-18)15-12-24(34)30(22)2/h8-9,16-18,20,33H,3-7,10-15H2,1-2H3,(H,27,28,29)
InChi Key
WELBJLUKWAJOQV-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
SKU | CAYM-37402-5 |
---|---|
Supplier Part Number | 37402-5 |
UM | EA |
UNSPSC | 12352200 |
Manufacturer | Cayman |
Temperature | -20 |
Refrigerated-Frozen | Refrigerated |
ProductLine | CAYM |
Qty | 5 |
MinOrderQty | 1 |
Weight | 7.00 |
Lead Time | 2 Business Days |
Hazardous | N |
CAS Number | 5352-53-4 |