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Cayman Gsk3β (Phospho-Ser9) Tr-Fret Assay Kit
Cayman Gsk3β (Phospho-Ser9) Tr-Fret Assay Kit - CAYM (Additional S&H Or Hazmat Fees May Apply)
List Price
$6,174.00
Your Price
$6,174.00
HOW MUCH YOU SAVE:
0.00 %
| NETA PART: | CAYM-500251-4800 |
| MFG.PART: | 500251-4800 |
| UNSPSC: | 12352200 |
| Manufacturer: | Cayman |
Product Description
Glycopyrrolate is an antagonist of muscarinic acetylcholine receptors (mAChRs; Kis = 0.42, 1.77, 0.52, 0.78, and 1.29 nM for the M1-M5 receptors, respectively). It induces relaxation of precontracted isolated human bronchi when used at concentrations of 0.01, 0.1, or 1 µM. Glycopyrrolate reduces post-prandial gastric antral motility in dogs when administered at a dose of 0.01 mg/kg. It inhibits salivation in a rat model of sialorrhea induced by pilocarpine with an ED50 value of 0.74 µg/kg. Formulations containing glycopyrrolate have been used in the treatment of sialorrhea, peptic ulcers, and chronic obstructive pulmonary disease (COPD).
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
3-[(2-cyclo
CAS Number
596-51-0
Synonyms
- AHR 504
- NSC 250836
- NSC 251251
- NSC 251252
Molecular Formula
C19H28NO3 • Br
Formula Weight
398.3
Purity
≥95%
Formulation
A crystalline solid
Solubility
- DMF: 30 mg/ml
- DMSO: 30 mg/ml
- Ethanol: 30 mg/ml
- PBS (pH 7.2): 10 mg/ml
SMILES
O=C(OC1CC[N+](C)(C)C1)C(O)(C2=CC=CC=C2)C3CCCC3.[Br-]
InChi Code
InChI=1S/C19H28NO3.BrH/c1-20(2)13-12-17(14-20)23-18(21)19(22,16-10-6-7-11-16)15-8-4-3-5-9-15;/h3-5,8-9,16-17,22H,6-7,10-14H2,1-2H3;1H/q+1;/p-1
InChi Key
VPNYRYCIDCJBOM-UHFFFAOYSA-M
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
| SKU | CAYM-500251-4800 |
|---|---|
| Supplier Part Number | 500251-4800 |
| UM | EA |
| UNSPSC | 12352200 |
| Manufacturer | Cayman |
| Temperature | -80 |
| Refrigerated-Frozen | Frozen |
| CountryOfOrigin | US |
| ProductLine | CAYM |
| Qty | 4800 |
| MinOrderQty | 1 |
| Weight | 7.00 |
| Lead Time | 2 Business Days |
| Hazardous | N |