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Cayman NCP-biotin Peptide (non-cyclized)
Cayman NCP-biotin Peptide (non-cyclized) - CAYM (Additional S&H Or Hazmat Fees May Apply)
List Price
$219.00
Your Price
$219.00
HOW MUCH YOU SAVE:
0.00 %
NETA PART: | CAYM-40255-1 |
MFG.PART: | 40255-1 |
UNSPSC: | 12352202 |
Manufacturer: | Cayman |
Product Description
PZM21 is a μ-opioid receptor agonist (Ki = 1.1 nM). It is selective for μ- over κ- and δ-opioid receptors (Kis = 18 and 506 nM, respectively). PZM21 induces Gi/o signaling (EC50 = 4.6 nM in HEK293T cells expressing human receptors) but has no detectable activity in a β-arrestin2 recruitment assay. In vivo, PZM21 (10, 20, and 40 mg/kg) induces analgesia in the hot plate test and reduces formalin-induced paw licking in mice when administered at a dose of 40 mg/kg.
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
N-[(2S)-2-(di methylamino)- 3-(4-hydroxy phenyl)propyl]- N-[(1S)-1-methyl- 2-(3-thienyl) ethyl]-urea
CAS Number
1997387-43-5
Molecular Formula
C19H27N3O2S
Formula Weight
361.5
Purity
≥95%
Formulation
A crystalline solid
Solubility
- DMF: 10 mg/ml
- DMSO: 1 mg/ml
- Ethanol: 10 mg/ml
- Ethanol:PBS (pH 7.2) (1:4): 0.2 mg/ml
λmax
229, 281 nm
SMILES
OC1=CC=C(C[C@H](N(C)C)CNC(N[C@@H](C)CC2=CSC=C2)=O)C=C1
InChi Code
InChI=1S/C19H27N3O2S/c1-14(10-16-8-9-25-13-16)21-19(24)20-12-17(22(2)3)11-15-4-6-18(23)7-5-15/h4-9,13-14,17,23H,10-12H2,1-3H3,(H2,20,21,24)/t14-,17-/m0/s1
InChi Key
MEDBIJOVZJEMBI-YOEHRIQHSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
SKU | CAYM-40255-1 |
---|---|
Supplier Part Number | 40255-1 |
UM | EA |
UNSPSC | 12352202 |
Manufacturer | Cayman |
MSDS URL | https://www.caymanchem.com/msdss/40255m.pdf |
Temperature | -20 |
Refrigerated-Frozen | Refrigerated |
CountryOfOrigin | US |
ProductLine | CAYM |
Qty | 1 |
MinOrderQty | 1 |
Weight | 7.00 |
Lead Time | 2 Business Days |
Hazardous | N |