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Cayman Aspartate Aminotransferase Colorimetric Activity Assay Kit
Cayman Aspartate Aminotransferase Colorimetric Activity Assay Kit; Size- 96 Wells; - CAYM (Additional S&H Or Hazmat Fees May Apply)
List Price
$291.00
Your Price
$291.00
HOW MUCH YOU SAVE:
0.00 %
NETA PART: | CAYM-701640-96 |
MFG.PART: | 701640-96 |
UNSPSC: | 41116104 |
Manufacturer: | Cayman |
Product Description
In humans, two forms of diacylglycerol lipase, DAGLα and DAGLβ, generate the endocannabinoid 2-arachidonoyl glycerol (2-AG; Item No. ) by attacking DAG at the sn-1 position. LEI-106 is a potent in vitro inhibitor of sn-1 DAGLα (IC50 = 18 nM). It blocks the hydrolysis of sn-1-oleoyl-2-AG, the natural substrate of DAGLα, with a Ki value of 0.7 µM. LEI-106 inhibits the hydrolysis of 2-AG by the monoacylglycerol lipase ABHD6 in mouse brain membrane homogenates and in HEK293T cell membrane preparations (Ki = 0.8 µM).
WARNING This product is not for human or veterinary use.
Technical Information
Formal Name
N-[(3,4- dihydro- 2,2-dimethyl- 2H-1- benzopyran- 6-yl) sulfonyl]-N- [(4-phenoxy phenyl) methyl]- glycine
CAS Number
1620582-23-1
Molecular Formula
C26H27NO6S
Formula Weight
481.6
Purity
≥98%
Formulation
A crystalline solid
Solubility
- DMF: 50 mg/ml
- DMF:PBS (pH 7.2) (1:1): 0.5 mg/ml
- DMSO: 30 mg/ml
- Ethanol: 0.1 mg/ml
λmax
245 nm
SMILES
OC(CN(S(C1=CC=C(OC(C)(C)CC2)C2=C1)(=O)=O)CC(C=C3)=CC=C3OC4=CC=CC=C4)=O
InChi Code
InChI=1S/C26H27NO6S/c1-26(2)15-14-20-16-23(12-13-24(20)33-26)34(30,31)27(18-25(28)29)17-19-8-10-22(11-9-19)32-21-6-4-3-5-7-21/h3-13,16H,14-15,17-18H2,1-2H3,(H,28,29)
InChi Key
FOEGBOXMDBPYEV-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room Temperature in continental US; may vary elsewhere
Stability
≥ 4 years
SKU | CAYM-701640-96 |
---|---|
Supplier Part Number | 701640-96 |
UM | EA |
UNSPSC | 41116104 |
Manufacturer | Cayman |
MSDS URL | https://www.caymanchem.com/msdss/701640m.pdf |
Temperature | -20 |
Refrigerated-Frozen | Refrigerated |
CountryOfOrigin | US |
ProductLine | CAYM |
Qty | 1 |
MinOrderQty | 1 |
Weight | 7.00 |
Lead Time | 2 Business Days |
Hazardous | N |